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B
MOLECULAR TARGETUniProt: P25021

HRH2

histamine receptor H2

75 compounds · BiohacksAI corpus v20260307-01

75
compounds
Compounds
75
Gene Symbol
HRH2
NCBI Gene
3274

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About HRH2

HRH2 (histamine receptor H2) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 75 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View HRH2 on UniProt →
Compounds Targeting HRH2 (50)
1
Tamoxifen
5.88
confidence
2
Clozapine
5.81
confidence
3
Imatinib
5.47
confidence
4
Risperidone
4.89
confidence
5
Quinacrine
4.63
confidence
6
Thioridazine
4.52
confidence
7
Amiodarone
4.51
confidence
8
Clomipramine
4.28
confidence
9
Promazine
4.19
confidence
10
Gentian Violet
4.03
confidence
11
Loperamide
3.93
confidence
12
Fluphenazine
3.91
confidence
13
Doxepin
3.50
confidence
14
Ketotifen
3.47
confidence
15
Desloratadine
3.26
confidence
300
studies
3.18
confidence
17
Imiquimod
3.14
confidence
18
Orphenadrine
2.94
confidence
19
Cimetidineorganic
0
studies
2.89
confidence
20
Ebastine
2.64
confidence
21
Clemastine
2.56
confidence
22
Dicyclomine
2.56
confidence
23
Bay 293
2.48
confidence
24
Latrepirdine
2.40
confidence
25
Penfluridol
2.40
confidence
26
Nantenine
2.08
confidence
27
Dexchlorpheniramine
1.95
confidence
28
Bay 876
1.95
confidence
29
Borussertib
1.95
confidence
297
studies
1.79
confidence
31
A 349821
1.79
confidence
32
Tirilazad
1.79
confidence
33
4 Methylhistamine
1.79
confidence
237
studies
1.61
confidence
299
studies
1.10
confidence
299
studies
1.10
confidence
300
studies
1.10
confidence
300
studies
1.10
confidence
299
studies
1.10
confidence
1000
studies
0.69
confidence
1000
studies
0.69
confidence
299
studies
0.69
confidence
994
studies
0.69
confidence
299
studies
0.69
confidence
259
studies
0.69
confidence
298
studies
0.69
confidence
280
studies
0.69
confidence
109
studies
0.69
confidence
299
studies
0.69
confidence
296
studies
0.69
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.