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B
MOLECULAR TARGETUniProt: P10721

KIT

KIT proto-oncogene, receptor tyrosine kinase

83 compounds · BiohacksAI corpus v20260307-01

83
compounds
Compounds
83
Gene Symbol
KIT
NCBI Gene
3815

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About KIT

KIT (KIT proto-oncogene, receptor tyrosine kinase) is a biological target studied in biomedical research. The BiohacksAI corpus identifies 83 compounds with documented interactions with this target, based on BindingDB assay data and PubMed literature.

View KIT on UniProt →
Compounds Targeting KIT (50)
1
Gefitinib
5.67
confidence
2
Erlotinib
5.55
confidence
3
Imatinib
5.47
confidence
4
Alvocidib
4.52
confidence
5
Cabozantinib
4.39
confidence
6
Foretinib
4.34
confidence
7
Tozasertib
4.33
confidence
8
Vandetanib
4.30
confidence
9
Ponatinib
4.26
confidence
10
Ruxolitinib
4.23
confidence
11
Ceritinib
4.19
confidence
12
Nilotinib
4.17
confidence
300
studies
4.17
confidence
14
Bosutinib
4.08
confidence
15
Doramapimod
4.06
confidence
16
Quizartinib
3.99
confidence
17
Semaxanib
3.93
confidence
18
Midostaurin
3.85
confidence
19
Brigatinib
3.81
confidence
20
Pazopanib
3.69
confidence
21
Vatalanib
3.69
confidence
300
studies
3.66
confidence
23
Nintedanib
3.61
confidence
24
Regorafenib
3.56
confidence
25
Canertinib
3.53
confidence
26
Tae 684
3.43
confidence
27
Pexidartinib
3.43
confidence
28
Fedratinib
3.40
confidence
29
Bms 777607
3.37
confidence
30
Linifanib
3.33
confidence
31
Saracatinib
3.33
confidence
298
studies
3.22
confidence
33
Tandutinib
3.22
confidence
34
Dovitinib
3.09
confidence
35
Jnj 7706621
3.09
confidence
36
Dasatinib Anhydrous
3.09
confidence
37
Lestaurtinib
3.04
confidence
38
Ruboxistaurin
2.94
confidence
39
Danusertib
2.94
confidence
40
Defosbarasertib
2.89
confidence
41
Barasertib
2.89
confidence
246
studies
2.83
confidence
43
R 406
2.83
confidence
44
Cediranib
2.83
confidence
45
Milciclib
2.77
confidence
46
Infigratinib
2.77
confidence
47
Masitinib
2.77
confidence
48
Pha 665752
2.71
confidence
49
Plx 4720
2.71
confidence
50
Enmd 2076
2.71
confidence
Top 50 compounds by confidence score. Derived from BindingDB assay data.
Data Source
Corpusv20260307-01
SourceBindingDB · ChEMBL · PubMed

All data is computationally derived from published research. Not medical advice. Independent validation required.